Metronidazole

Metronidazole

Class: Nitroimidazole.Mol weight: 171First used in 1960. Mechanism of action: Metronidazole enters the susceptible (bacterial/parasite) cells by passive diffusion. It gets activated to a nitroso compound which causes oxidative damage to the DNA. It also inhibits DNA repair. The conversion of metronidazole to nitroso compound creates a concentration gradient, and more metronidazole enters the cells. The aerobic bacteria lack the necessary…

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Tigecycline

Tigecycline

Nature: Glycylcycline, a member of the tetracycline family. Semisynthetic derivative of minocycline.MW: 585.6 Mechanism of action: 1. Bind to 30S ribosomal subunit and inhibit protein synthesis – It inhibits the attachment of aminoacyl tRNA to the A site and prevents chain elongation, i.e. block the translation process.2. Inhibit mitochondrial protein synthesis by binding to 70…

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Rotavirus vaccine (study note)

Vaccine Efficacy– Protect against gastroenteritis due to rotavirus serotypes G1P, G2P, G3P, G4P, and G9P; some efficacy against uncommon rotavirus genotypes G8P and G12P.– Over 85% effective at protecting against severe rotavirus gastroenteritis in the first two years of life. Administration of the vaccine Rotarix® should not be given to infants under 6 weeks of age.WHO recommends infants should…

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Fusidic acid

Fusidic acid

Fusidic acid was discovered in Copenhagen, Denmark and introduced to clinical practice in the 1960s.It was derived from a fungus, Fusidium coccineum. Fusidic acid has a structural similarity with the steroid molecule. You can see in the picture the molecular structure is similar to prednisolone. For this reason, it is called a steroid antibiotic. It also…

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Norovirus

Epidemiology Norovirus is the most common cause of epidemic gastroenteritis worldwide. In the UK, norovirus outbreak is usually seen in the winter months. The virus Norovirus is a small non-enveloped RNA virus of the caliciviridae family. It has ten genogroups, but I, II and IV are primarily implicated in human infection. Genogroup II is most…

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ceftolozane tazobactam

Ceftolozane-tazobactam

Class: 5th generation cephalosporin.Available as ceftolozane-tazobactam, a beta lactam-beta lactamase inhibitor (BLBLI) combination. Mechanism of Action: Similar to other beta-lactam antibiotics. It binds to the penicillin-binding protein (PBP) to inhibit the biosynthesis of the cell wall.It binds with the PBP3 of E coli and PBP3, PBP1a, and PBP1b of Pseudomonas aeruginosa. Mechanism of resistance: It is…

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